A Novel Approach of Formulation & Evaluation of Tablet in Capsule Device for GI Protection Pain Management
Abstract
This research article presents a novel approach in the formulation and evaluation of a tablet in capsule device aimed at providing GI protection and effective pain management. Key aspects include the development of Aceclofenac Extended-Release tablets and Misoprostol Immediate Release tablets, enclosed in a hard gelatin capsule. The study…
Dissolution enhancement of a model poorly water-soluble drug, atorvastatin, with ordered mesoporous…
13. December 2015 The purpose of this study was to develop mesoporous silica materials incorporated with poorly water-soluble drug atorvastatin calcium (AC) in order to…
Role of Polymeric Excipients in the Stabilization of Olanzapine when Exposed to Aqueous Environments
13. December 2015 Maria Paisana 1, MartinWahl 2 and João Pinto 1,*Received: 5…
Optimizing Semisolid Dosage Forms
13. December 2015 Quality by design, in-vitro release testing, and modern analytical methods are improving understanding and control of these complex formulations. Years…
Assessing Drug-Excipient Interactions in the Formulation of Isoniazid Tablets
12. December 2015 Wagner Wollinger,*,a Raphael A. da Silva,b Andréa B. da…
Folic acid loaded lipid nanocarriers with promoted skin antiaging and antioxidant efficacy
09. December 2015 Aging is the progressive deterioration of physiological functions in organisms. Folic acid (FA) can be used as antiaging. The objective of this research is…
Risperidone oral disintegrating mini-tablets: A robust-product for pediatrics
09. December 2015 Risperidone oral disintegrating mini-tablets: A robust-product for pediatrics…
Development of oral dispersible tablets containing prednisolone nanoparticles for the management of…
09. December 2015 Yi-Dan Chen,1 Zhong-Yuan Liang,1 Yan-Yan Cen,1 He Zhang,2…
Background review for sodium laurilsulfate used as an excipient – EMA draft report
08. December 2015 Background review for sodium laurilsulfate used as an excipient…
Potentially harmful excipients in neonatal medicines: a pan-European observational study
Objective: We aimed to describe administration of eight potentially harmful excipients of interest (EOI)-parabens, polysorbate 80, propylene glycol, benzoates, saccharin sodium, sorbitol, ethanol and benzalkonium chloride-to…
Myrrh a traditional medicine or a multipurpose pharmaceutical excipient
08. December 2015 Fatemeh Erfanfar1, 2, Hashem Montaseri1, 3,*, Abdolali…
Fluid bed film coating of fine ibuprofen particles
08. December 2015 Highlights • Geldart group C ibuprofen particles were silica dry coated to enable fluidization. • Aeration testing and flow function…
Use of Polyvinyl Alcohol as a Solubility-Enhancing Polymer for Poorly Water Soluble Drug Delivery…
08. December 2015 Polyvinyl alcohol (PVAL) has not been investigated in a binary formulation as a concentration-enhancing polymer owing to its high melting point/high…
INFLUENCE OF IONIC STRENGTH ON THE RHEOLOGICAL PROPERTIESOF HYDROXYPROPYLMETHYL…
07. December 2015 Jaroslav M. Katona*, Alena Tomšik, Sandra Dj. Bučko and Lidija…
Role of excipients and polymeric advancements in preparation of floating drug delivery systems
07. December 2015 Int J Pharm Investig. 2015 Jan-Mar; 5(1): 1–12.doi:…
Advanced stable lipid-based formulations for a patient-centric product design
07. December 2015 Multiparticulate dosage forms are a recent strategy to meet the special needs of children, elderly people and patients suffering from dysphagia. Our study…
IMPACT OF EXCIPIENT VARIABILITY ON DRUG PRODUCT PROCESSING AND PERFORMANCE
07. December 2015 It is rare to have a pharmaceutical dosage form presented with just the pure active pharmaceutical ingredient because the drug substance does not possess…
Improved oral absorption of tacrolimus by a solid dispersion with hypromellose and sodium lauryl…
06. December 2015 A novel surfactant-incorporated hydroxypropyl methylcellulose (HPMC) solid dispersion (SD) system was constructed in order to facilitate the release rate…
Dissolution of Danazol Amorphous Solid Dispersions: Supersaturation and Phase Behavior as a Function…
06. December 2015 Amorphous solid dispersions (ASDs) are of great interest as enabling formulations because of their ability to increase the bioavailability of poorly…
Development and Evaluation of Liquid and Solid Self-Emulsifying Drug Delivery Systems for…
06. December 2015 Anna Czajkowska-Kośnik 1,*, Marta Szekalska 1, Aleksandra…
Improving oral drug bioavailability with polycations?
06. December 2015 The administration of drugs via the oral route is challenging due to the (bio)chemical aggressivity of the digestive system and to the presence of barriers…
Extended-release venlafaxine pellets: scaling up – Poster Ashland AAPS 2014
06. December 2015
Introduction:
This study from Ashland was undertaken to investigeate the influence of coating process scale when applying an organic solvent based modified release coating to multiparticulates using a Wurster…
Impact of moisture and magnesium stearate functionality on manufacturability of wet granulated…
05. December 2015 During the development of a wet granulated 850 mg metformin hydrochloride tablet formulation, the tablets exhibited high friability (>3% w/w)…
A novel floating controlled release drug delivery system prepared by hot-melt extrusion
05. December 2015 Floating dosage forms are an important formulation strategy for drugs with a narrow absorption window and low intestinal solubility, and for localized…
Evaluation of formulation and effects of process parameters on drug release and mechanical…
05. December 2015 Nenad D. Nikolić1, Djordje P. Medarević2, Svetlana R. Ibrić2,…
An Overview on Polymethacrylate Polymers in Gastroretentive Dosage Forms
05. December 2015 An Overview on Polymethacrylate Polymers in Gastroretentive DosageForms…
Fluidized Bed Processing
04. December 2015 TTC Workshop January 26-28, 2016 in Binzen / Germany This workshop on fluidized bed technology is a perfect combination of…
Quantifying effects of moisture content on flow properties of microcrystalline cellulose using a…
04. December 2015 Highlights • Flowability of Avicel PH102 significantly deteriorates with increasing RH (or moisture) • Powder density exhibits a maximum at an…
Collodial silica-induced hypersensitivity: myth or reality
03. December 2015 Background Many excipients have been reported to induce drug hypersensitivity (e.g. colouring additives, preservatives). Colloidal silica has never been…
Optimization of pantoprazole enteric coated pellets by QbD
03. December 2015 Optimization of pantoprazole enteric coated pellets by QbD OPTIMIZATION OF…
Combination of bubble liposomes and ultrasound for gene delivery
02. December 2015 pharmaceutics-07-00344.pdf…
Study on Topical Ocular Delivery System of Certain Non-steroidal Anti-inflammatory Drugs
30. November 2015 5366-10508-1-SM.pdf…
Development of curcumin floating tablets based on low density foam powder
30. November 2015
The floating drug delivery system (FDDS) has become an increasingly attractive system for gastroretentive dosage forms because it can prolong gastric retention time and improve drug bioavailability . Using…
Microemulsion-based hydrogels of itraconazole: evaluation of characteristics and stability
30. November 2015 Itraconazole (ITZ) is a broad spectrum triazole antifungal drug and commercially available as oral forms. However, effective topical forms are interesting…
Effect of precipitation/re-dissolution processes from the supersaturated solution on the intestinal…
30. November 2015 Effect of precipitation/re-dissolution processes from the supersaturated solution on the intestinal absorption of poorly water-soluble drugs As one of the…